Detalles de la búsqueda
1.
Uncovering the Power of GPR18 Signalling: How RvD2 and Other Ligands Could Have the Potential to Modulate and Resolve Inflammation in Various Health Disorders.
Molecules
; 29(6)2024 Mar 12.
Artículo
Inglés
| MEDLINE | ID: mdl-38542895
2.
Anti-inflammatory effects of new human histamine H3 receptor ligands with flavonoid structure on BV-2 neuroinflammation.
Inflamm Res
; 72(2): 181-194, 2023 Feb.
Artículo
Inglés
| MEDLINE | ID: mdl-36370200
3.
Evaluation of Some Safety Parameters of Dual Histamine H3 and Sigma-2 Receptor Ligands with Anti-Obesity Potential.
Int J Mol Sci
; 24(8)2023 Apr 19.
Artículo
Inglés
| MEDLINE | ID: mdl-37108661
4.
The Potent and Selective Histamine H3 Receptor Antagonist E169 Counteracts Cognitive Deficits and Mitigates Disturbances in the PI3K/AKT/GSK-3ß Signaling Pathway in MK801-Induced Amnesia in Mice.
Int J Mol Sci
; 24(16)2023 Aug 12.
Artículo
Inglés
| MEDLINE | ID: mdl-37628900
5.
Novel GPR18 Ligands in Rodent Pharmacological Tests: Effects on Mood, Pain, and Eating Disorders.
Int J Mol Sci
; 24(10)2023 May 20.
Artículo
Inglés
| MEDLINE | ID: mdl-37240392
6.
Antiplatelet Effects of Selected Xanthine-Based Adenosine A2A and A2B Receptor Antagonists Determined in Rat Blood.
Int J Mol Sci
; 24(17)2023 Aug 29.
Artículo
Inglés
| MEDLINE | ID: mdl-37686188
7.
Anti-Inflammatory Activities of 8-Benzylaminoxanthines Showing High Adenosine A2A and Dual A1/A2A Receptor Affinity.
Int J Mol Sci
; 24(18)2023 Sep 05.
Artículo
Inglés
| MEDLINE | ID: mdl-37762006
8.
Multitargeting Histamine H3 Receptor Ligands among Acetyl- and Propionyl-Phenoxyalkyl Derivatives.
Molecules
; 28(5)2023 Mar 03.
Artículo
Inglés
| MEDLINE | ID: mdl-36903593
9.
Trisubstituted 1,3,5-Triazines as Histamine H4 Receptor Antagonists with Promising Activity In Vivo.
Molecules
; 28(10)2023 May 19.
Artículo
Inglés
| MEDLINE | ID: mdl-37241939
10.
Structure Prediction, Evaluation, and Validation of GPR18 Lipid Receptor Using Free Programs.
Int J Mol Sci
; 23(14)2022 Jul 18.
Artículo
Inglés
| MEDLINE | ID: mdl-35887268
11.
GPR18-Mediated Relaxation of Human Isolated Pulmonary Arteries.
Int J Mol Sci
; 23(3)2022 Jan 26.
Artículo
Inglés
| MEDLINE | ID: mdl-35163351
12.
Preliminary Evidence of the Potent and Selective Adenosine A2B Receptor Antagonist PSB-603 in Reducing Obesity and Some of Its Associated Metabolic Disorders in Mice.
Int J Mol Sci
; 23(21)2022 Nov 03.
Artículo
Inglés
| MEDLINE | ID: mdl-36362227
13.
KSK-74: Dual Histamine H3 and Sigma-2 Receptor Ligand with Anti-Obesity Potential.
Int J Mol Sci
; 23(13)2022 Jun 24.
Artículo
Inglés
| MEDLINE | ID: mdl-35806019
14.
Benzophenone Derivatives with Histamine H3 Receptor Affinity and Cholinesterase Inhibitory Potency as Multitarget-Directed Ligands for Possible Therapy of Alzheimer's Disease.
Molecules
; 28(1)2022 Dec 28.
Artículo
Inglés
| MEDLINE | ID: mdl-36615435
15.
An insight into the structure of 5-spiro aromatic derivatives of imidazolidine-2,4-dione, a new group of very potent inhibitors of tumor multidrug resistance in T-lymphoma cells.
Bioorg Chem
; 109: 104735, 2021 04.
Artículo
Inglés
| MEDLINE | ID: mdl-33640632
16.
Cyanobiphenyls: Novel H3 receptor ligands with cholinesterase and MAO B inhibitory activity as multitarget compounds for potential treatment of Alzheimer's disease.
Bioorg Chem
; 114: 105129, 2021 09.
Artículo
Inglés
| MEDLINE | ID: mdl-34217977
17.
The Structural Determinants for α1-Adrenergic/Serotonin Receptors Activity among Phenylpiperazine-Hydantoin Derivatives.
Molecules
; 26(22)2021 Nov 20.
Artículo
Inglés
| MEDLINE | ID: mdl-34834117
18.
Discovery of Potential, Dual-Active Histamine H3 Receptor Ligands with Combined Antioxidant Properties.
Molecules
; 26(8)2021 Apr 15.
Artículo
Inglés
| MEDLINE | ID: mdl-33921144
19.
Biphenylalkoxyamine Derivatives-Histamine H3 Receptor Ligands with Butyrylcholinesterase Inhibitory Activity.
Molecules
; 26(12)2021 Jun 11.
Artículo
Inglés
| MEDLINE | ID: mdl-34208297
20.
In silico and in vitro studies on interaction of novel non-imidazole histamine H3R antagonists with CYP3A4.
Bioorg Med Chem Lett
; 30(11): 127147, 2020 06 01.
Artículo
Inglés
| MEDLINE | ID: mdl-32249114